Protheine inhibitor ke karoloana e kopanang le catalyst, e sitisang ketso ea eona. Li-Catalysts, e leng liprotheine tse thusang likarabo tsa motsoako ka ho sa feleng, li sebetsa ka phetoho ea likaroloana tsa substrate ho ba lihlahisoa.[1] K'hemik'hale e finyella sena ka ho thibela substrate sebakeng sa eona se matla, sebaka se itseng se potlakisang mohato o boima ka ho fetisisa oa karabo.


Protheine inhibitor e kenella potolohong ena ka e 'ngoe kapa e' ngoe e thibelang sebaka se matla sa lik'hemik'hale, ho boloka substrate ho thibela, kapa ho thibela sebaka se seng hape holim'a motsoako, ho nyahamisa catalyst's catalysis ea karabo. Li-inhibitors li ka bonts'a lithibelo tse ka khutlisoang kapa tse ke keng tsa khutlisoa. Li-inhibitors tse sa khoneheng li etsa tlamahano ea motsoako le protheine, e e hatelle ho fihlela tlamo e robeha. 


Ka lehlakoreng le leng, li-reversible inhibitors li tlama ka mokhoa o sa kopane 'me li ka ikarola hang-hang ho tsoa ho li-catalyst, tsa lumella protheine ho tsoela pele ka bokhoni ba eona. Ho ipapisitsoe le hore na ba ikopanya le lik'hemik'hale, motsoako oa motsoako oa motsoako, kapa ka bobeli, li-reversible inhibitors li baka mefuta e fapaneng ea thibelo.


Li-inhibitors

0
  • Vismodegib

    Nomoro ea CAS: 879085-55-9
    Ponahalo: Ho tsoa phofo e tšoeu kapa e Yellow kapa Crystal
    Standard: ka tlung
    Kopo: Anti tumor; anti-mofetshe 
    Matla a Phepelo: 50kg ka khoeli
    Ho hloeka: ≥99%
    Tefo: T/T, LC kapa DA
    Nako ea ho Thomelloa: Setoko se Itokisitseng ka har'a Warehouse ea Lehae, matsatsi a 1-3
    Origin: China
    Ho romella: DHL, FedEx, TNT, EMS, Ka Leoatle, Ka Moea
    Ha e khone ho rekisetsa batho ka bomong
  • Verteporfin API

    Nomoro ea CAS: 129497-78-5
    Ponahalo: Botala bo lefifi ho isa ho botsho bo tiileng
    Standard: ka tlung
    Kopo: Patlisiso ea Lab 
    Matla a Phepelo: 100g ka khoeli
    Ho hloeka: ≥96%
    Tefo: T/T, LC kapa DA
    Nako ea ho Thomelloa: Setoko se Itokisitseng ka har'a Warehouse ea Lehae, matsatsi a 1-3
    Origin: China
    Ho romella: DHL, FedEx, TNT, EMS, Ka Leoatle, Ka Moea
    Ha e khone ho rekisetsa batho ka bomong
  • EPZ-6438

    Nomoro ea CAS: 1403254-99-8
    Ponahalo: Phofo ea kristale e tšoeu kapa e bosoeu
    Standard: ka tlung
    Kopo: Patlisiso ea Lab  
    Matla a Phepelo: 1000g ka khoeli
    Ho hloeka: ≥98%
    Tefo: T/T, LC kapa DA
    Nako ea ho Thomelloa: Setoko se Itokisitseng ka har'a Warehouse ea Lehae, matsatsi a 1-3
    Origin: China
    Ho romella: DHL, FedEx, TNT, EMS, Ka Leoatle, Ka Moea
    Ha e khone ho rekisetsa batho ka bomong
  • Alagebrium Chloride

    Nomoro ea CAS: 341028-37-3
    Ponahalo: phofo e batlang e le tšoeu kapa e tšoeu e mebala
    Standard: ka tlung
    Matla a Phepelo: 1000g ka khoeli
    Ho hloeka: ≥99%
    Tefo: T/T, LC kapa DA
    Nako ea ho Thomelloa: Setoko se Itokisitseng ka har'a Warehouse ea Lehae, matsatsi a 1-3
    Origin: China
    Ho romella: DHL, FedEx, TNT, EMS, Ka Leoatle, Ka Moea
    Ha e khone ho rekisetsa batho ka bomong
  • AZD 1480

    Nomoro ea CAS: 935666-88-9
    Ponahalo: e tšoeu ho ea ho beige phofo
    Standard: ka tlung
    Matla a Phepelo: 1000g ka khoeli
    Ho hloeka: ≥99%
    Tefo: T/T, LC kapa DA
    Nako ea ho Thomelloa: Setoko se Itokisitseng ka har'a Warehouse ea Lehae, matsatsi a 1-3
    Origin: China
    Ho romella: DHL, FedEx, TNT, EMS, Ka Leoatle, Ka Moea
    Ha e khone ho rekisetsa batho ka bomong
  • AZD 8055

    Nomoro ea CAS: 1009298-09-2
    Ponahalo: Bosehla bo kganyang ho isa ho bosehla bo tiileng
    Standard: ka tlung
    Matla a Phepelo: 1000g ka khoeli
    Ho hloeka: ≥99%
    Tefo: T/T, LC kapa DA
    Nako ea ho Thomelloa: Setoko se Itokisitseng ka har'a Warehouse ea Lehae, matsatsi a 1-3
    Origin: China
    Ho romella: DHL, FedEx, TNT, EMS, Ka Leoatle, Ka Moea
    Ha e khone ho rekisetsa batho ka bomong
  • Clascoterone phofo

    Nomoro ea CAS: 19608-29-8
    Ponahalo: phofo e tšoeu ho isa ho e mosehla
    Standard: ka tlung
    Matla a Phepelo: 100kg ka khoeli
    Ho hloeka: ≥99%
    Tefo: T/T, LC kapa DA
    Nako ea ho Thomelloa: Setoko se Itokisitseng ka har'a Warehouse ea Lehae, matsatsi a 1-3
    Origin: China
    Ho romella: DHL, FedEx, TNT, EMS, Ka Leoatle, Ka Moea
    Ha e khone ho rekisetsa batho ka bomong
  • Setipiprant phofo

    Nomoro ea CAS: 866460-33-5
    Ponahalo: phofo e mosehla e bobebe
    Standard: ka tlung
    Matla a Phepelo: 1000g ka khoeli
    Ho hloeka: ≥99%
    Tefo: T/T, LC kapa DA
    Nako ea ho Thomelloa: Setoko se Itokisitseng ka har'a Warehouse ea Lehae, matsatsi a 1-3
    Origin: China
    Ho romella: DHL, FedEx, TNT, EMS, Ka Leoatle, Ka Moea
    Ha e khone ho rekisetsa batho ka bomong
  • Pyrilutamide

    Nomoro ea CAS: 1272719-00-2
    Ponahalo: phofo e tšoeu ho isa ho e mosehla
    Standard: ka tlung
    Matla a Phepelo: 1000g ka khoeli
    Ho hloeka: ≥99%
    Tefo: T/T, LC kapa DA
    Nako ea ho Thomelloa: Setoko se Itokisitseng ka har'a Warehouse ea Lehae, matsatsi a 1-3
    Origin: China
    Ho romella: DHL, FedEx, TNT, EMS, Ka Leoatle, Ka Moea
    Ha e khone ho rekisetsa batho ka bomong
  • Finerenone API

    Nomoro ea CAS: 1050477-31-0
    Ponahalo: Phofo ea kristale e tšoeu ho ea ho mosehla
    Standard: ka tlung
    Matla a Phepelo: 5000g ka khoeli
    Ho hloeka: ≥99%
    Tefo: T/T, LC kapa DA
    Nako ea ho Thomelloa: Setoko se Itokisitseng ka har'a Warehouse ea Lehae, matsatsi a 1-3
    Origin: China
    Ho romella: DHL, FedEx, TNT, EMS, Ka Leoatle, Ka Moea
    Ha e khone ho rekisetsa batho ka bomong
  • Glecaprevir

    CAS: 1365970-03-1
    Ponahalo: Phofo e tšoeu ho ea ho Off-White
    Assay: 98%
    Lebitso: YIHUI
    Ho paka: 1g; 10g; 100g
    Matla a Phepelo: 2000g ka khoeliShelf Life: Lilemo tse peli
    Kopo: lipatlisiso tsa laboratori
    Tefo: T/T, LC kapa DA
    Mohlala: e teng
    Nako ea thomello: Setoko se Itokisitseng ka har'a Warehouse ea Lehae, matsatsi a 1-3
    Kapele-pele le ho Sireletsa Thomello
    Origin: China
    Thomello: DHL,FedEx,TNT,EMS,Ka Leoatle,Ka Moea
    Setifikeiti: ISO9001, ISO22000, HACCP, HALAL, KOSHER
    Ha e khone ho rekisetsa batho ka bomong
  • EA-408-RTA

    CAS: 1474034-05-3
    Ponahalo: Phofo e soeufetse
    Assay: 98%
    Lebitso: YIHUI
    Ho paka: 1g; 10g; 100g
    Matla a Phepelo: 2000g ka khoeli
    Shelf Life: Lilemo tse peli
    Kopo: lipatlisiso tsa laboratori
    Tefo: T/T, LC kapa DA
    Mohlala: e teng
    Nako ea thomello: Setoko se Itokisitseng ka har'a Warehouse ea Lehae, matsatsi a 1-3
    Kapele-pele le ho Sireletsa Thomello
    Origin: China
    Thomello: DHL,FedEx,TNT,EMS,Ka Leoatle,Ka Moea
    Setifikeiti: ISO9001, ISO22000, HACCP, HALAL, KOSHER
    Ha e khone ho rekisetsa batho ka bomong
27