Protheine inhibitor ke karoloana e kopanang le catalyst, e sitisang ketso ea eona. Li-Catalysts, e leng liprotheine tse thusang likarabo tsa motsoako ka ho sa feleng, li sebetsa ka phetoho ea likaroloana tsa substrate ho ba lihlahisoa.[1] K'hemik'hale e finyella sena ka ho thibela substrate sebakeng sa eona se matla, sebaka se itseng se potlakisang mohato o boima ka ho fetisisa oa karabo.
Protheine inhibitor e kenella potolohong ena ka e 'ngoe kapa e' ngoe e thibelang sebaka se matla sa lik'hemik'hale, ho boloka substrate ho thibela, kapa ho thibela sebaka se seng hape holim'a motsoako, ho nyahamisa catalyst's catalysis ea karabo. Li-inhibitors li ka bonts'a lithibelo tse ka khutlisoang kapa tse ke keng tsa khutlisoa. Li-inhibitors tse sa khoneheng li etsa tlamahano ea motsoako le protheine, e e hatelle ho fihlela tlamo e robeha.
Ka lehlakoreng le leng, li-reversible inhibitors li tlama ka mokhoa o sa kopane 'me li ka ikarola hang-hang ho tsoa ho li-catalyst, tsa lumella protheine ho tsoela pele ka bokhoni ba eona. Ho ipapisitsoe le hore na ba ikopanya le lik'hemik'hale, motsoako oa motsoako oa motsoako, kapa ka bobeli, li-reversible inhibitors li baka mefuta e fapaneng ea thibelo.
Li-inhibitors
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Vismodegib
Nomoro ea CAS: 879085-55-9
Ponahalo: Ho tsoa phofo e tšoeu kapa e Yellow kapa Crystal
Standard: ka tlung
Kopo: Anti tumor; anti-mofetshe
Matla a Phepelo: 50kg ka khoeli
Ho hloeka: ≥99%
Tefo: T/T, LC kapa DA
Nako ea ho Thomelloa: Setoko se Itokisitseng ka har'a Warehouse ea Lehae, matsatsi a 1-3
Origin: China
Ho romella: DHL, FedEx, TNT, EMS, Ka Leoatle, Ka Moea
Ha e khone ho rekisetsa batho ka bomong -
Verteporfin API
Nomoro ea CAS: 129497-78-5
Ponahalo: Botala bo lefifi ho isa ho botsho bo tiileng
Standard: ka tlung
Kopo: Patlisiso ea Lab
Matla a Phepelo: 100g ka khoeli
Ho hloeka: ≥96%
Tefo: T/T, LC kapa DA
Nako ea ho Thomelloa: Setoko se Itokisitseng ka har'a Warehouse ea Lehae, matsatsi a 1-3
Origin: China
Ho romella: DHL, FedEx, TNT, EMS, Ka Leoatle, Ka Moea
Ha e khone ho rekisetsa batho ka bomong -
EPZ-6438
Nomoro ea CAS: 1403254-99-8
Ponahalo: Phofo ea kristale e tšoeu kapa e bosoeu
Standard: ka tlung
Kopo: Patlisiso ea Lab
Matla a Phepelo: 1000g ka khoeli
Ho hloeka: ≥98%
Tefo: T/T, LC kapa DA
Nako ea ho Thomelloa: Setoko se Itokisitseng ka har'a Warehouse ea Lehae, matsatsi a 1-3
Origin: China
Ho romella: DHL, FedEx, TNT, EMS, Ka Leoatle, Ka Moea
Ha e khone ho rekisetsa batho ka bomong -
Alagebrium Chloride
Nomoro ea CAS: 341028-37-3
Ponahalo: phofo e batlang e le tšoeu kapa e tšoeu e mebala
Standard: ka tlung
Matla a Phepelo: 1000g ka khoeli
Ho hloeka: ≥99%
Tefo: T/T, LC kapa DA
Nako ea ho Thomelloa: Setoko se Itokisitseng ka har'a Warehouse ea Lehae, matsatsi a 1-3
Origin: China
Ho romella: DHL, FedEx, TNT, EMS, Ka Leoatle, Ka Moea
Ha e khone ho rekisetsa batho ka bomong -
AZD 1480
Nomoro ea CAS: 935666-88-9
Ponahalo: e tšoeu ho ea ho beige phofo
Standard: ka tlung
Matla a Phepelo: 1000g ka khoeli
Ho hloeka: ≥99%
Tefo: T/T, LC kapa DA
Nako ea ho Thomelloa: Setoko se Itokisitseng ka har'a Warehouse ea Lehae, matsatsi a 1-3
Origin: China
Ho romella: DHL, FedEx, TNT, EMS, Ka Leoatle, Ka Moea
Ha e khone ho rekisetsa batho ka bomong -
AZD 8055
Nomoro ea CAS: 1009298-09-2
Ponahalo: Bosehla bo kganyang ho isa ho bosehla bo tiileng
Standard: ka tlung
Matla a Phepelo: 1000g ka khoeli
Ho hloeka: ≥99%
Tefo: T/T, LC kapa DA
Nako ea ho Thomelloa: Setoko se Itokisitseng ka har'a Warehouse ea Lehae, matsatsi a 1-3
Origin: China
Ho romella: DHL, FedEx, TNT, EMS, Ka Leoatle, Ka Moea
Ha e khone ho rekisetsa batho ka bomong -
Clascoterone phofo
Nomoro ea CAS: 19608-29-8
Ponahalo: phofo e tšoeu ho isa ho e mosehla
Standard: ka tlung
Matla a Phepelo: 100kg ka khoeli
Ho hloeka: ≥99%
Tefo: T/T, LC kapa DA
Nako ea ho Thomelloa: Setoko se Itokisitseng ka har'a Warehouse ea Lehae, matsatsi a 1-3
Origin: China
Ho romella: DHL, FedEx, TNT, EMS, Ka Leoatle, Ka Moea
Ha e khone ho rekisetsa batho ka bomong -
Setipiprant phofo
Nomoro ea CAS: 866460-33-5
Ponahalo: phofo e mosehla e bobebe
Standard: ka tlung
Matla a Phepelo: 1000g ka khoeli
Ho hloeka: ≥99%
Tefo: T/T, LC kapa DA
Nako ea ho Thomelloa: Setoko se Itokisitseng ka har'a Warehouse ea Lehae, matsatsi a 1-3
Origin: China
Ho romella: DHL, FedEx, TNT, EMS, Ka Leoatle, Ka Moea
Ha e khone ho rekisetsa batho ka bomong -
Pyrilutamide
Nomoro ea CAS: 1272719-00-2
Ponahalo: phofo e tšoeu ho isa ho e mosehla
Standard: ka tlung
Matla a Phepelo: 1000g ka khoeli
Ho hloeka: ≥99%
Tefo: T/T, LC kapa DA
Nako ea ho Thomelloa: Setoko se Itokisitseng ka har'a Warehouse ea Lehae, matsatsi a 1-3
Origin: China
Ho romella: DHL, FedEx, TNT, EMS, Ka Leoatle, Ka Moea
Ha e khone ho rekisetsa batho ka bomong -
Finerenone API
Nomoro ea CAS: 1050477-31-0
Ponahalo: Phofo ea kristale e tšoeu ho ea ho mosehla
Standard: ka tlung
Matla a Phepelo: 5000g ka khoeli
Ho hloeka: ≥99%
Tefo: T/T, LC kapa DA
Nako ea ho Thomelloa: Setoko se Itokisitseng ka har'a Warehouse ea Lehae, matsatsi a 1-3
Origin: China
Ho romella: DHL, FedEx, TNT, EMS, Ka Leoatle, Ka Moea
Ha e khone ho rekisetsa batho ka bomong -
Glecaprevir
CAS: 1365970-03-1
Ponahalo: Phofo e tšoeu ho ea ho Off-White
Assay: 98%
Lebitso: YIHUI
Ho paka: 1g; 10g; 100g
Matla a Phepelo: 2000g ka khoeliShelf Life: Lilemo tse peli
Kopo: lipatlisiso tsa laboratori
Tefo: T/T, LC kapa DA
Mohlala: e teng
Nako ea thomello: Setoko se Itokisitseng ka har'a Warehouse ea Lehae, matsatsi a 1-3
Kapele-pele le ho Sireletsa Thomello
Origin: China
Thomello: DHL,FedEx,TNT,EMS,Ka Leoatle,Ka Moea
Setifikeiti: ISO9001, ISO22000, HACCP, HALAL, KOSHER
Ha e khone ho rekisetsa batho ka bomong -
EA-408-RTA
CAS: 1474034-05-3
Ponahalo: Phofo e soeufetse
Assay: 98%
Lebitso: YIHUI
Ho paka: 1g; 10g; 100g
Matla a Phepelo: 2000g ka khoeli
Shelf Life: Lilemo tse peli
Kopo: lipatlisiso tsa laboratori
Tefo: T/T, LC kapa DA
Mohlala: e teng
Nako ea thomello: Setoko se Itokisitseng ka har'a Warehouse ea Lehae, matsatsi a 1-3
Kapele-pele le ho Sireletsa Thomello
Origin: China
Thomello: DHL,FedEx,TNT,EMS,Ka Leoatle,Ka Moea
Setifikeiti: ISO9001, ISO22000, HACCP, HALAL, KOSHER
Ha e khone ho rekisetsa batho ka bomong
