Actinomycin D
NAKO ea CAS: 50-76-0
MOQ: 1g
Assay: 99%
Lebitso: YIHUI
Ho paka: 1g; 10g; 100g
Matla a Phepelo: 1000g ka khoeli
E sebelisitsoeng: Lik'hemik'hale tsa Laboratori
Nako ea thomello:e fumaneha
Shelf Life: Lilemo tse peli
Ha e khone ho rekisetsa batho ka bomong
- Phano e potlakileng
- boleng tiisetsa
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Product Introduction
Actinomycin D ke eng?
Actinomycin D, eo hape e tsejoang e le Dactinomycin kapa Actinomycin, ke e 'ngoe ea lithibela-mafu tsa bohlokoa ka ho fetisisa tsa peptide sehlopheng sa actinomycin se insulated ho tloha Streptomyces bacteria set up insoil.Ke haholo hygroscopic brilliant red crystalline powder eo butle-butle e lahleheloang ke ho sebetsa ha e pepesehetse leseli. E ne e le e 'ngoe ea li-agent tsa pele tsa chemotherapeutic,' me esale e sebelisoa ka nako e telele. E ne e le moriana oa pele oa lithibela-mafu o nang le thepa e thibelang mofetše ho sibolloa ke batho. SelmanA. Waksman le mosebetsimmoho le yena H.B. Woodruff o ile a e fumana ka lekhetlo la pele ka 1940. Dactinomycin e ile ea kenngoa kopong ea Merck tlas'a lebitso la Cosmegen ka mor'a ho fuoa tumello ke American FDA ka la 10 Tšitoe, 1964. e bontšitsoe lithutong tsa baeloji ea cellular ho hatella recap. E na le bokhoni ba ho hokahana le DNA setsing sa ho qala bocha, ho etsa motsoako o nang le DNA le ho qhekella bokhoni ba RNA polymerase ba ho kopanya RNA. E na le bokhoni ba ho tlama DNA e nang le likarolo tse peli, e lumellang hore e hatelle sehlahisoa sa RNA ho phaella tabeng ea ho ba le tšusumetso ho phetisetso ea DNA. ho ntse ho le joalo, bo-rasaense ka kakaretso ba sebelisa litšitiso tse itseng tsa ho ikatisa ha DNA, tse tšoanang le tsa hydroxyurea, tse loketseng tšebeliso ea laboratori. Ha ho etsoa lipatlisiso tse kenyelletsang cytometry ea ho phalla le ho ithuta ka lisele tsa bitsy, phofo ea Actinomycin D le limela tsa eona tsa fluorescent, 7- aminoactinomycin D (7- AAD), li sebelisoa e le litšila.
Li loketse hantle bakeng sa ho ngola DNA ka lebaka la kamano ea tsona le likarolo tsa GC-rich DNA. Kaha 7-AAD e ka ikamahanya le DNA e nang le mela e le 'ngoe, e boetse e na le molemo bakeng sa ho shebella cell apoptosis le ho bolella lisele tse phelang ntle le tse shoeleng.
Information Basic
Lebitso la sehlahisoa: Actinomycin D
Lebitso le leng: Actinomycin D, Actinomycin IV, Actinomycin C1, Dactinomycin;Actactinomycin A IV;actinomycin7;actinomycinaiv
CAS:50-76-0
MF:C62H86N12O16
MW: 1255.42
EINECS: 246-818-3
Qhibiliha ntlha: 251-253 ℃
Solubility: ethanol, DMSO: E tsitsitse ka har'a litharollo tse nang le metsi ho 2-8 ℃.
mocheso oa polokelo. 2-8℃
Botsitso: E tsitsitseng
Mokhoa o raliloeng:

Tekanyetso ea boleng
Items | songolo | Results |
Ponahalo | Kristale e bofubelu bo khanyang kapa bo bofubelu ba lamunu kapa phofo, hoo e batlang e se na monko; ha ho na bopaki bo bonahalang ba ho silafatsoa ke ntho e tsoang kantle ho naha | Liphetoho |
Boitsebiso | Leqhubu le phahameng la absorptive ke 241nm le 442 nm. Karolelano ea ho monya ho 241nm le 442 nm ke 1.3 ~ 1.5 Sephetho sa UV se lumellana le maemo | Liphetoho
Liphetoho |
Ho lahleheloa ke ho omisoa | NMT 5.0% | 3.0% |
Ho potoloha ho itseng | -292°~-317° | -314 ° |
Li-solvents tsa nakoana | Acetone NMT 5000ppm Ethanol NMT 5000ppm Ethanol acetate NMT 5000ppm THF NMT 720ppm Toluene NMT 890ppm | 700ppm 1600ppm 1350ppm 230ppm 370ppm |
Lintho tse amanang | RRT 1.18 ~ 1.20 RRT 1.26 ~ 1.27 Kakaretso ea litšila NMT 4.0% | 0.5% 1.6% 3.2% |
Boemo ba Endotoxin | ≤100EU/mg | 78EU/mg |
Assay (ka ho omisa) | 95.0% ~ 103.0% | 95.8% |
Polokelo: boloka sebakeng se omileng. | ||
Qetello: sehlahisoa se kopana le maemo a USP. | ||
mosebetsi
Actinomycin D e na le litlamorao tse ngata:
Sethibela-mafu sa mofetše:Sethibela-mafu sa pele se nang le litšobotsi tse thibelang mofetše se tla fumanoa ke batho ke actinomycin D. E tlama DNA le ho thibela RNA polymerase ho hlahisa RNA, ho thibela lisele tsa excrescence hore li se ke tsa ata le ho ata.
Phello e khahlanong le ho ruruha: e na le tšusumetso e khahlanong le ho ruruha ka ho thibela likarabo tsa bofetoheli le ts'ebetso ea tsamaiso e tlokotsing. Sena se theola tokollo ea baemeli ba borabele le ho fokotsa matšoao a amanang le ho ruruha le tšenyo ea lithaole.
Immunosuppressive effect: e na le tšusumetso ea ho itšireletsa mafung ka ho fokotsa ho ata le ho sebetsa ha lisele tse tlokotsing le ho thibela bokhoni ba tsamaiso e tlokotsing ea ho hlahisa masole a 'mele. Ka pheko ea immunosuppressive kamora ho fetisoa ha setho, e ea sebelisoa.
Antiviral effect: e na le thepa ea antiviral e etsang hore e sebetse khahlanong le likokoana-hloko tse itseng. E ka emisa ho ata le ho ata ha livaerase.
Antibacterial effect: e na le ketso ea antibacteria e sebetsang khahlanong le likokoana-hloko tse ling. E na le bokhoni ba ho thibela kholo ea baktheria le ho fokotseha.
Ho bohlokoa ho hlakisa hore Ke sethethefatsi sa bohlokoa 'me se lokela ho sebelisoa feela tlas'a tlhokomelo ea croaker le ka hloko. Ho netefatsa polokeho le katleho, lozenge le mokhoa oa tsamaiso li lokela ho khethoa ho latela maemo a ikhethang.
kopo
Likopo tsa Dactinomycin kenyeletsa:
Phekolo e khahlanong le mofetše:Mokhahlelo oa pele oa chemotherapy drug actinomycin D o lula o sebelisoa maemong a bongaka ho phekola mefuta e mengata ea mofetše o mobe, ho kenyeletsoa le makhopho a matla a bana, Wilms excrescence, rhabdomyosarcoma le hepatocellular melanoma.
Phekolo ea Immunosuppressive: e sebelisoa phekong ea immunosuppressive kamora ho fetisoa ha setho sa 'mele hobane e na le bokhoni ba ho thibela sistimi e tlokotsing. E eketsa sekhahla sa katleho ea transplantation le ho thusa ho theola karabelo ea ho hana litho tse fanoeng.
Mafu a ho ruruha: ke litekanyetso tse thibelang ho ruruha li e etsa hore e tšoanelehe bakeng sa phekolo ea maemo a mang a hlohlelletsang matla, ho akarelletsa le ramatiki ea ramatiki le tletlebo ea mala a seditious.
Ho bohlokoa ho tseba hore E ka baka litlamorao tse mpe joalo ka ho se sebetse hantle ha sebete, mathata a mala, le khatello ea moko oa masapo. Ka hona, pele ho kalafo Actinomycin-d, litsebi tsa bongaka li hlahloba matšoao a mokuli le ho etsa mekhoa e khethehileng ea phekolo ho itšetlehile ka boemo ba bona bo ikhethang. Ho bohlokoa ho sebelisa Actinomycin D tlas'a tlhokomelo ea ngaka le ho ela hloko likhothaletso tsa bona le mehato ea ts'ireletso.
Botsitso le polokelo
Ho tsitsisa le ho boloka maemo a eona ke a latelang:
Mocheso oa polokelo: Ho boloka botsitso ba eona, e lokela ho bolokoa mochesong o batang (-20 degrees Celsius). E ka nkoa e bolokoa ka mocheso o tlase le ho feta bakeng sa polokelo ea nako e telele, joalo ka -80 degrees Celsius.
Tshireletso ya kganya: e lokela ho bolokoa maemong a e sireletsang kganyeng le ho dula ntle le letsatsi le otlolohileng ka lebaka la kutlo ya yona kganyeng. Ho fokotsa matla a khanya ea moriana, lijana tse opaque kapa tse lefifi li ka sebelisoa ho boloka.
Tikoloho e omileng: Ho boloka mongobo o se ke oa ama moriana, o lokela ho bolokoa sebakeng se omileng. Ho etsa bonnete ba hore moriana o omme, ho ka sebelisoa lijana tse tiisitsoeng kapa thepa ea ho paka.
Qoba lipotoloho tsa ho qhibiliha ha leqhoa: e ka 'na ea se ke ea tsitsa ka makhetlo a mangata a ho qhibiliha, kahoo ho molemo ho qoba ho etsa joalo hangata pele o sebelisoa.
Ka kopo hlokomela seo Actinomycin dmso e lokela ho bolokoa maemong a boletsoeng ka holimo ho boloka botsitso le katleho ea eona. Hlahloba chebahalo ea moriana le letsatsi la ho felloa ke nako pele o sebelisoa.
Ho paka le ho tsamaisa ka sekepe
itokisa: 1kg / mokotla oa foil; 5kg / carton; 25kg / fiber drum; kapa ho paka joalo ka kopo ea hau.
Tlhophiso:Letšoao le ikhethileng; sephutheloana se ikhethileng; Ho etsa litšoantšo
Ho tsamaisa ka sekepe:
Item | bongata | Nako ea ETA | Mokhoa oa ho Romela |
E ngotsoe ke Courier | Kg50kg | 7-15days | Fedex, DHL, UPS, TNT, EMS joalo-joalo. E potlakile ebile e bonolo |
Ka Moea | 50kg ~ 200kg | 3-5days | Ka potlako le ka theko e tlaase |
Haufi le Leoatle | Bongata bo boholo | 20-35days | Tsela e theko e tlaase |
Nako ea ho etella pele: Matsatsing a 3 a mosebetsi ka mor'a ho fumana tefo.
tefo Nako
Ke Hobane'ng ha U Khetha Xi'an Yihui?
Tlhaloso ea bareki
Litifikeiti tsa Xi'an Yihui
Feme ea Xi'an Yihui le Botoro
Melemo ea Rōna
Phihlelo e ruileng: re na le Lilemo tse 13 tsa boiphihlelo ba litsebi;
Bareki lefatšeng ka bophara: rekisetsa linaha tse fetang 100;
Fana ka lihlahisoa tse fapa-fapaneng: lihlahisoa li sebelisitsoe ho mefuta eohle e meholo ea machaba lefapheng la lithethefatsi, lijo tsa lijo, litlolo, phepo ea liphoofolo le lijo tse sebetsang hantle.
Theko esale pele: MOQ e tlase ka theko ea tlholisano;
Setifikeiti sa boleng: ISO; Halal; Kosher e netefalitsoe
Tšebeletso ea ka mor'a thekiso: Sehlopha sa litsebi 7 * lihora tse 24 custotšebeletso ea ka.
Ha re phethela
Ka kakaretso, joalo ka setsebi Actinomycin D moetsi, re na le thekenoloji e tsoetseng pele, melemo e mengata, boleng bo holimo, boiphihlelo bo bongata ba tlhahiso, le lits'ebeletso tse ntle haholo. Melemo ena e tla etsa hore Dactinomycin ea rona e hlahelle tlholisanong ea 'maraka le ho hapa tšepo le tšehetso ea bareki. ha o hloka Actinomycin D phofo, pls ikutloe u lokolohile ho ikopanya le rona neng kapa neng. re tla u araba kapele.
lintlha tsa rona tsa ho ikopanya:
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