Acarbose API

Lebitso la Sehlahisoa: Acarbose
Origin: China
Matla a Phepelo: 1ton ka khoeli
Mohlala o Teng: E
Shelf Life: Lilemo tse peli
Tefo: T/T, LC kapa DA
Setifikeiti: ISO9001, ISO22000, HACCP, HALAL, KOSHER
Teko ea Motho oa Boraro: e fumaneha
Plant Audition: e fumaneha
Ha e khone ho rekisetsa batho ka bomong
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Product Introduction

Mofani oa Acarbose API

Khamphani ea Xi'an Yihui ke moetsi ea hloahloa oa Acarbose. Re ka hlahisa Acarbose e nang le litaba tsa 99.9%. E ka sebelisoa lijong, meriana, linthong tsa tlhokomelo ea bophelo, kapa lihlahisoa tsa litlolo, 'me ea kopana le litekanyetso tsa USP, BP, EP, CP. Re ka u fa lihlahisoa tsa boleng bo phahameng ka ho fetesisa ka litefiso tsa tlholisano. Khetho ea hau e ntle ka ho fetisisa bakeng sa morekisi ea hloekileng oa Acarbose ke Khamphani ea Xi'an Yihui!

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Acarbose API ke eng?

Acarbose API, motsoako oa manyolo o nang le foromo ea lik'hemik'hale C25H43NO18 le CAS No. 56180-94-0.Ke phofo e tšoeu kapa e tšoeu, e kang crystalline, ha e na monko, e baba hanyenyane, e qhibilihang metsing. Lebitso la lik'hemik'hale la acarbose ke 4, 6-o-ethyl mannitol-keto-alpha-d-glucose.

Acarbose API ke motsoako o sebetsang oa lithethefatsi tsa alpha-glucosidase inhibitor, hangata tse hlahisoang indastering ka ho belisoa ha likokoana-hloko, tse kang actinomyces. Ts'ebetso ea tlhahiso haholo-holo e kenyelletsa setso sa likokoana-hloko, ho itšehla thajana le ho itlhoekisa, karabelo ea phepelo ea li-reactor le ho ntšoa, karohano ea sehlahisoa le tlhoekiso, le mehato e meng, eo karabelo ea phepelo ea reactor e leng mohato oa mantlha oa ho lokisa carboxylate ho tsoa ho tsoekere. E sebelisoa haholo ho phekola lefu la tsoekere la mofuta oa 2.


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Information Basic

Ponahalo

phofo e tšoeu kapa e mosehla, amorphous

Moralo oa mohaho

Molecular Formula

C25H43NO18

Ntlha e qhibilihisang

165 ho isa ho 170 ℃

 CAS 56180-94-0.webp

Boima ba 'mele

645.61

Sebaka se belang

971.6 ℃

CAS No.

56180-94-0

segokanyipalo

1.74 g/cm³

Ho hloeka

mets 98%

nako ea ho boloka.

Mocheso oa kamore.

Tekanyetso ea boleng

Items

songolo

Results

litlhaku

E tšoeu kapa e mosehla, phofo ea amorphous, hygroscopic. E qhibiliha haholo ka metsing, e qhibiliha ka methanol, hoo e batlang e sa qhibilihe ka har'a methylene chloride

Liphetoho

Boitsebiso

Joalo ka EP10.0

Liphetoho

Ho monya

Max. 0.15 ho 425nm bakeng sa tharollo S.

0.001

Tlhahlobo (ka anhydrousbasis)

95.0% ~ 102.0%

99.3%

metsi

≤4.0%

1.8%

Potoloho e khethehileng ea optical

+168°~+183°

+ 181 °

Molora o sulfated

≤0.2%

0.06%

PH

5.5 ~ 7.5

6.6

Lisebelisoa tse boima

≤20ppm

Liphetoho


               


               


               

Ntho e amanang le yona

Tšilafalo A Max 0.6%

0.2%

Tšilafalo B Max 0.5%

0.2%

Tšilafalo C Max 1.5%

0.2%

Impurity D Max 1.0%

0.3%

Impurity E Max 0.2%

a fosahetseng

Tšilafalo F Max 0.3%

a fosahetseng

Impurity G Max 0.3%

a fosahetseng

Tšilafalo efe kapa efe e 'ngoe e litšila Ke 0.2%

Liphetoho

Kakaretso ea litšila Max 3.0%

1.1%

Qetello: sehlahisoa sena se lumellana le litlhaloso tsa EP10.0.

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Acarbose e sebelisetsoa eng?

Acarbose API ke sethethefatsi se tsebahalang se sebelisoang haholo ho alafa lefu la tsoekere la mofuta oa 2. Haholo-holo, e khetholloa e le letlotlo la nascence-glucosidase 'me e sebetsa ka mala a manyenyane ho fokotsa ho senyeha le ho qoelisoa ha lik'habohaedreite. Setlhare sena ka kakaretso se hlalosoa e le tlatsetso ea lijo le boikoetliso 'me hangata se sebelisoa hammoho le mefuta e meng ea lefu la tsoekere.

e sebetsa ka ho thibela li-enzyme tseo ka tloaelo li senyang lik'habohaedreite tse rarahaneng hore e be tsoekere e bonolo, e tšoanang le ea glucose. Ka ho theola tšilo ea lijo le ho qoelisoa ha tsoekere ena, e thusa ho laola maemo a tsoekere ea mali ho batho ba nang le lefu la tsoekere. Sena se ka thusa ho thusa mathata le ho lokisa mathata a bophelo bo botle.

Ntle le ho alafa lefu la tsoekere la mofuta oa 2, e boetse e ithutoe bakeng sa tšebeliso ea eona e felletseng ho fokotsa tšokelo ea litletlebo tsa pelo le mathata a mang a pelo. Liphuputso tse ling li bontšitse hore moriana ona o ka thusa ho ntlafatsa lipid biographies le ho fokotsa ho ruruha 'meleng, e leng se ka lebisang ho fokotseng tšokelo ea litletlebo tsa pelo ha nako e ntse e ea.

Tšebeliso e 'ngoe ea eona e hlakileng e ka kenyelletsa kalafo ea maemo a mang a amanang le ho hanyetsa insulin, a tšoanang le polycystic ovary pattern(PCOS) le metabolic pattern. ho ntse ho le joalo, ho hlokahala lipatlisiso tse eketsehileng pele litšebeliso tsena tse hlakileng li ka utloisisoa ka botlalo.

Ka kakaretso, ke setlhare sa bohlokoa bakeng sa kalafo ea lefu la tsoekere la mofuta oa 2 le maemo a mang a amanang le ona. Ka ho fokotsa ho qoelisoa ka lik'habohaedreite le ho thusa ho laola maemo a tsoekere ea mali, sethethefatsi sena se ka thusa ho fokotsa tšokelo ea mathata le ho ntlafatsa liphello tsa bophelo bo botle ka kakaretso. Leha ho le joalo, bua le croaker ea hau mabapi le hore na e ka ba khetho e ntle ea kalafo ho uena, Haeba u fumanoe u e-na le lefu la tsoekere la mofuta oa 2 kapa boemo bo bong bo amanang le bona.

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ho lokisetsa

Mokhoa oa ho kopanya oa Acarbose e ka akaretsoa ka mehato e meraro e latelang:

  1. Synthesis ea aminocyclitol: Sedoheptulose-7-phosphate e na le letoto la likarabo tsa enzymatic tse kenyeletsang intramolecular cyclization, epimerization, dehydrogenation, dehumidification, phosphorylation, le nucleotidylation ho hlahisa NDP-1-epi-valienol-7-phosphate.

  2. Motsoako oa 4-amino-4,6-dideoxyglucose:D- glucose-1-phosphate e fetoloa dTDP ka nucleotidylation, dehumidification, le transamination.

  3. Synthesis of acarviosyl moiety: NDP-1-epi-valienol-7-phosphate le dTDP li utloa bohloko karabelo ea phetisetso ea tsoekere e lipakeng tsa glycosyltransferase ho etsa dTDP- acarbose-7-phosphate, eo hape e kopanang ka kotloloho le maltose ho etsa hore acarbose-7-phosphate. Acarbose-7-phosphate e entsoe ka har'a sele, empa hore qetellong e hlahise acarbose, e hloka ho tsamaisoa ka ntle ho sele ka transmembrane protein AcbWXY/GacWXY ebe e etsoa dephosphorylation.

Litlamorao ke life bakeng sa Acarbose?

Acarbose ke setlhare se sebelisoang ho phekola lefu la tsoekere la mofuta oa 2. Le hoja sethethefatsi sena se sebetsa hantle ho laola maemo a tsoekere ea mali, se boetse se na le thepa e 'maloa e fanoeng e ka' nang ea ama linyeoe. Tse ling tsa tse atileng ka ho fetisisa lehlakoreng thepa ea Acarbose e thibelang botsofali li boletsoe ka tlase

1. Mathata a ka mpeng: E ​​ka tsoala ho ruruha, khase le letšollo. Mathata ana a tšilo ea lijo a ka ba a tšoenyang haholo-holo ho batho ba kileng ba sebetsana le mathata a mala.

2. Tsoekere e tlaase maling: E ​​ka tsoala hypoglycemia, e khetholloang ka maemo a tlase a tsoekere maling. Linyeoe tse noang moriana ona li lokela ho tšoha matšoao le matšoao a hypoglycemia, 'me li lokela ho ja lijo tse tloaelehileng, tse leka-lekaneng ho qoba litlamorao tsena.

3. Mathata a sebete: E ka baka tšenyo ea sebete maemong a sa tloaelehang. Linyeoe tse noang moriana ona li lokela ho ba le ts'ebetso ea sebete ea tsona kamehla.

4. Lekhopho la letlalo: Maemo a mang a ka hlaha lekhopho ha le ntse le le noa. Le hoja letšoao lena hangata le le bobebe, linyeoe li lokela ho tsebisa batho ba nang le croaker haeba ba bona liphetoho tse ncha kapa tse sa tloaelehang tsa letlalo.

5. Boitšoaro ba ho kula: Maemo a mang a ka paka karabelo e sa rateheng ho acarbose. Matšoao a ka kenyelletsa bothata ba ho hema, ho hema ka thata, kapa ho ruruha ha sefahleho le 'metso. Linyeoe li lokela ho batla thuso ea bongaka ka mokhoa o sa tsitsang haeba li bona leha e le efe ea matšoao ana.

6. Flatulence: Ho tsebahala hore ho baka moea o mongata kapa ho tsoa ha khase. Letšoao lena le ka tšoenya bakuli ba bang empa hangata ha le kotsi.
7. Ho kena-kenana le ho kenngoa ha limatlafatsi: E ka 'na ea kena-kenana le ho kenngoa ha limatlafatsi tse itseng, tse kang k'halsiamo le vithamine D. Bakuli ba noang meriana ena ba lokela ho ja lijo tse nang le limatlafatsi tsena kapa ba nke tlatsetso ho qoba mefokolo.
Ho bohlokoa hore bakuli ba noang acarbose ba ele hloko litla-morao tsena tse ka bang teng le ho buisana le ngaka ea bona ka mathata afe kapa afe. Haeba leha e le efe ea matšoao ana e e-ba matla kapa a phehella, bakuli ba lokela ho ea ngakeng hang-hang. Ka kakaretso, acarbose ke moriana o thusang ho laola maemo a tsoekere ea mali ho bakuli ba nang le lefu la tsoekere la mofuta oa 2, empa ho bohlokoa ho ela hloko litlamorao tse ka bang teng.

Ho paka le ho tsamaisa ka sekepe

itokisa: 1kg / mokotla oa foil; 5kg / lebokose; 25kg / moropa oa fiber; kapa ho paka joalo ka kopo ea hau.

Tlhophiso: Letšoao le ikhethileng; Sephutheloana se ikhethileng; Graphic customization

Ho tsamaisa ka sekepe:

Item

bongata

Nako ea ETA

Mokhoa oa ho Romela

E ngotsoe ke Courier

Kg50kg

7-15days

Fedex, DHL, UPS, TNT, EMS joalo-joalo.

E potlakile ebile e bonolo

Ka Moea

50kg ~ 200kg

3-5days

Ka potlako le ka theko e tlaase

Haufi le Leoatle

Bongata bo boholo

20-35days

Tsela e theko e tlaase

Nako ea ho etella pele: Matsatsing a 3 a mosebetsi ka mor'a ho fumana tefo.

tefo Nako

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Ke Hobane'ng ha U Khetha Xi'an Yihui?

Tlhaloso ea bareki

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Litifikeiti tsa Xi'an Yihui

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Feme ea Xi'an Yihui le Botoro

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Melemo ea Rōna

Phihlelo e ruileng: re na le Lilemo tse 13 tsa boiphihlelo ba litsebi;

Bareki lefatšeng ka bophara: rekisetsa linaha tse fetang 100;

Fana ka lihlahisoa tse fapa-fapaneng: lihlahisoa li sebelisitsoe ho mefuta eohle e meholo ea machaba lefapheng la lithethefatsi, lijo tsa lijo, litlolo, phepo ea liphoofolo le lijo tse sebetsang hantle.

Theko esale pele: MOQ e tlase ka theko ea tlholisano;

Setifikeiti sa boleng: ISO; Halal; Kosher e netefalitsoe

Tšebeletso ea ka mor'a thekiso: Sehlopha sa litsebi lihora tse 7 * 24 tšebeletso ea bareki.

Ha re phethela

Ho akaretsa, Xi 'an Yihui Company e le setsebi sa moetsi oa Acarbose API , ka lihlahisoa tsa boleng bo phahameng, boemo bo phahameng ba lipatlisiso le bokhoni ba nts'etsopele, lisebelisoa tse tsoetseng pele tsa tlhahiso le theknoloji, tšebeletso e phethahetseng ka mor'a thekiso le melemo e meng, ke khetho ea bareki ea molekane ea loketseng.

haeba u e hloka, pls ikutloe u lokolohile ho ikopanya le rona neng kapa neng. re tla u araba ASAP.

Lintlha tsa rona tsa ho ikopanya:

E-mail: sales@yihuipharm.com
Tel: 0086-29-89695240
WeChat kapa WhatsApp: 0086-17792415937

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